• 3-Chloro-N′-(2-hydroxybenzylidene) benzohydrazide: An LSD1-Selective Inhibitor and Iron-Chelating Agent for Anticancer Therapy 

      Sarno, Federica; Papulino, Chiara; Franci, Gianluigi; Andersen, Jeanette hammer; Cautain, Bastien; Melardo, Colombina; Altucci, Lucia; Nebbioso, Angela; Andersen, Jeanette H. (Journal article; Tidsskriftartikkel; Peer reviewed, 2018-09-07)
      Despite the discovery and development of novel therapies, cancer is still a leading cause of death worldwide. In order to grow, tumor cells require large quantities of nutrients involved in metabolic processes, and an increase in iron levels is known to contribute to cancer proliferation. Iron plays an important role in the active site of a number of proteins involved in energy metabolism, DNA ...